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Library · Digestive & liver · Anti-inflammatory and digestive system regulation

VIP (Vasoactive Intestinal Peptide)

Vasoactive Intestinal Polypeptide, VIP-28, Aviptadil

Vasoactive Intestinal Peptide is a natural 28-amino-acid hormone involved in digestion, immune regulation, and neurological function, acting as a potent vasodilator and anti-inflammatory. Its synthetic form, Aviptadil, has been studied for conditions including respiratory distress and holds Orphan Drug status for pulmonary arterial hypertension, available via compounding pharmacies.

Research score 80/100. Reference only, not a dose.

  • Anti-inflammatory
  • Gut Health
  • Immune Boosting
  • Inflammation Resolution
  • Neuroprotection
  • Cardioprotection
US status
Research Chemical / Compounded Medication
Approval
Not FDA approved as a drug. Has Orphan Drug Designation for pulmonary arterial hypertension.
Evidence
Human studies for various conditions including chronic inflammatory response syndrome (CIRS), with ongoing research for diabetes and PCOS.
Research score
80 / 100
Indication
Investigational - Inflammatory Conditions, Diabetes, PCOS
Origin
USA
Source category
Digestive System
Status group
Research chemical

Mechanism

Binds VPAC1/VPAC2 receptors to raise cAMP and activate PKA, suppressing pro-inflammatory cytokines while boosting anti-inflammatory IL-10; relaxes gut smooth muscle and regulates intestinal secretion and barrier integrity, and shows neuroprotective effects via PI3K/Akt while dampening NF-κB-driven inflammation in immune cells.

Safety file

Generally considered safe, particularly as a compounded nasal spray.

  • Flushing
  • Hypotension
  • Diarrhea
  • Nausea
  • Dizziness